07. Risperidone and Paliperidone
Key Points
- For patients on oral risperidone, the active moiety level (risperidone level + 9-OH risperidone level), is exactly 7.0 times the oral dose.
- For CYP2D6 extensive metabolizers, the risperidone: 9-OH risperidone ratio is 0.2 with a range of 0.1 to 0.3.
- The clinical data from trials of Risperdal Consta or Invega Sustenna can be used to provide approximate oral risperidone dose equivalents.
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